(Q33408481)

26 July 2017

title

An AlphaScreen-based high-throughput screen to identify inhibitors of Hsp90-cochaperone interaction (English)

1 reference

26 July 2017

1 reference

26 July 2017

1 reference

26 July 2017

Christopher P Austin

1 reference

26 July 2017

Lynne Regan

1 reference

26 July 2017

Pingjun Zhu

1 reference

26 July 2017

Fang Yi

1 reference

26 July 2017

James Inglese

series ordinal

1 reference

26 July 2017

publication date

11 February 2009

1 reference

Journal of Biomolecular Screening

26 July 2017

language of work

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26 July 2017

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26 July 2017

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26 July 2017

page(s)

273-281

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A novel class of small molecule inhibitors of Hsp90.

26 July 2017

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3066041

The Hsp90 molecular chaperone: an open and shut case for treatment

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3066041

Inhibitors of the heat shock response: biology and pharmacology

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3066041

Heat shock protein 90: the cancer chaperone

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3066041

Phase I trial of 17-allylamino-17-demethoxygeldanamycin in patients with advanced cancer

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3066041

Phase I and pharmacodynamic study of 17-(allylamino)-17-demethoxygeldanamycin in adult patients with refractory advanced cancers

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3066041

A detergent-based assay for the detection of promiscuous inhibitors

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3066041

Quantitative high-throughput screening: a titration-based approach that efficiently identifies biological activities in large chemical libraries

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3066041

Functional specificity of co-chaperone interactions with Hsp90 client proteins.

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3066041

The Mechanism of Hsp90 regulation by the protein kinase-specific cochaperone p50(cdc37)

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3066041

14 July 2018

What is a co-chaperone?

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3066041

A specific mechanism of nonspecific inhibition

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3066041

Ligand discrimination by TPR domains. Relevance and selectivity of EEVD-recognition in Hsp70 x Hop x Hsp90 complexes

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3066041

Structure of TPR domain-peptide complexes: critical elements in the assembly of the Hsp70-Hsp90 multichaperone machine

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3066041

Hop as an adaptor in the heat shock protein 70 (Hsp70) and hsp90 chaperone machinery

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3066041

The tetratricopeptide repeat domain of protein phosphatase 5 mediates binding to glucocorticoid receptor heterocomplexes and acts as a dominant negative mutant

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3066041

Luminescent oxygen channeling immunoassay: measurement of particle binding kinetics by chemiluminescence.

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3066041

A small molecule designed to bind to the adenine nucleotide pocket of Hsp90 causes Her2 degradation and the growth arrest and differentiation of breast cancer cells

14 July 2018

1 reference

Crossref

https://api.crossref.org/works/10.1177%2F1087057108330114

AlphaScreen kinase HTS platforms

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1177%2F1087057108330114

Phase I trial of 17-allylamino-17-demethoxygeldanamycin in patients with advanced cancer

21 January 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/19211782

12 December 2020

inferred from PubMed ID database lookup

A duplexed phenotypic screen for the simultaneous detection of inhibitors of the molecular chaperone heat shock protein 90 and modulators of cellular acetylation

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/19211782

12 December 2020

inferred from PubMed ID database lookup

Designed TPR modules as novel anticancer agents

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/19211782

12 December 2020

inferred from PubMed ID database lookup

Identifiers

DOI

10.1177/1087057108330114

1 reference

release_dinyx3rztrenpchc6u4bjh5jx4

26 July 2017

Fatcat ID

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/dinyx3rztrenpchc6u4bjh5jx4

24 November 2022

mapped directly with Wikidata item

PMC publication ID

3066041

1 reference

26 July 2017

1 reference