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Drug-target residence time: critical information for lead optimization.
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Europe PubMed Central
PMC publication ID
2918722
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20663707%20AND%20SRC:MED&resulttype=core&format=json
retrieved
8 February 2020
review article
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Europe PubMed Central
title
Drug-target residence time: critical information for lead optimization
(English)
1 reference
stated in
Europe PubMed Central
PMC publication ID
2918722
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20663707%20AND%20SRC:MED&resulttype=core&format=json
retrieved
8 February 2020
main subject
drug discovery
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author
Peter J. Tonge
series ordinal
2
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Europe PubMed Central
PMC publication ID
2918722
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20663707%20AND%20SRC:MED&resulttype=core&format=json
retrieved
8 February 2020
author name string
Hao Lu
series ordinal
1
1 reference
stated in
Europe PubMed Central
PMC publication ID
2918722
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20663707%20AND%20SRC:MED&resulttype=core&format=json
retrieved
8 February 2020
publication date
19 July 2010
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stated in
Europe PubMed Central
PMC publication ID
2918722
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20663707%20AND%20SRC:MED&resulttype=core&format=json
retrieved
8 February 2020
published in
Current Opinion in Chemical Biology
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stated in
Europe PubMed Central
PMC publication ID
2918722
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20663707%20AND%20SRC:MED&resulttype=core&format=json
retrieved
8 February 2020
volume
14
1 reference
stated in
Europe PubMed Central
PMC publication ID
2918722
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20663707%20AND%20SRC:MED&resulttype=core&format=json
retrieved
8 February 2020
issue
4
1 reference
stated in
Europe PubMed Central
PMC publication ID
2918722
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20663707%20AND%20SRC:MED&resulttype=core&format=json
retrieved
8 February 2020
page(s)
467-474
1 reference
stated in
Europe PubMed Central
PMC publication ID
2918722
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20663707%20AND%20SRC:MED&resulttype=core&format=json
retrieved
8 February 2020
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The dynamics of drug-target interactions: drug-target residence time and its impact on efficacy and safety
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Evaluation of enzyme inhibitors in drug discovery. A guide for medicinal chemists and pharmacologists
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The role of binding kinetics in therapeutically useful drug action
1 reference
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based on heuristic
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Identifiers
DOI
10.1016/J.CBPA.2010.06.176
1 reference
stated in
Europe PubMed Central
PMC publication ID
2918722
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20663707%20AND%20SRC:MED&resulttype=core&format=json
retrieved
8 February 2020
PMC publication ID
2918722
1 reference
stated in
Europe PubMed Central
PMC publication ID
2918722
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20663707%20AND%20SRC:MED&resulttype=core&format=json
retrieved
8 February 2020
PubMed publication ID
20663707
1 reference
stated in
Europe PubMed Central
PMC publication ID
2918722
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20663707%20AND%20SRC:MED&resulttype=core&format=json
retrieved
8 February 2020
ResearchGate publication ID
45388673
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